DigestAI news desk

Cut through the AI noise.

Research

Mirror-Score benchmarks D-peptide design tools against real-world affinity

Researchers introduced Mirror-Score, a new scoring method for evaluating D-peptide designs in drug discovery. The tool assesses heterochiral D-peptide/L-protein complexes and includes a public benchmark of 31 crystal structures from four target families, 18 with verified affinities. The study found that raw ProteinMPNN negative log-likelihood (NLL) rankings do not correlate with measured binding…

1 source primary source

Key points

  • Mirror-Score benchmarks 31 crystal structures, 18 with verified affinities across four target families
  • Raw ProteinMPNN NLL rankings show poor affinity correlation (Spearman 0.19) and vary by target
  • Boltz-2 cofolding confidence achieves 0.90 correlation for viral-entry targets but requires family-specific calibration

The authors emphasize that calibration must be target-family-specific due to limited cross-family transferability. They also outline a prospective design protocol for antimicrobial-resistance targets like Pseudomonas aeruginosa’s LasR and LecB, including mirrored structures and diffusion-model inputs. All code, data, and scripts are openly available on GitHub.

The story so far

2 episodes →
  1. Mirror-Score benchmarks D-peptide design tools against real-world affinitythis story
Read the original at arXiv cs.AI · by Jiada Li primary sourceOpen source ↗
Topics · follow one to build your own front page

The headline, key points and digest above were generated by Digest AI's editorial model from the linked sources. Automated summaries can contain errors: the sources are the record. Spotted a mistake? Tell us. Published by Martin K., who runs Digest AI and handles corrections.

Comments

via GitHub Discussions

More in Research

All →

Related stories